SCHEMBL537371

SCHEMBL537371

COc1c(N2CC3CCCNC3C2)ccc2c(=O)c3c(O)c(C#N)sc3n(C3CC3)c12

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KCNH2 Q12809 2/20 0.33
ALK Q9UM73 4/20 0.33
HTR3A P46098 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2675165 1.00 KDM4E (0.41) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL2674752 0.87 KDM4E (0.57) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL2675462 0.84 ALK (0.39) KCNH2ALK
SCHEMBL605159 0.82 KDM4E (0.41) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL2675766 0.79 KCNH2 (0.39) KCNH2ALK
SCHEMBL537747 0.78 IKBKB (0.33) ALK
SCHEMBL2676459 0.74 ALK (0.33) KDM4EALDH1A1HPGDHSD17B10ALK
SCHEMBL2676884 0.73 KDM4E (0.41) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL2880218 0.73 KDM4E (0.41) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL537639 0.72 IKBKB (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414368-A2 HYDROXYTHIENOQUINOLONES AND RELATED COMPOUNDS AS ANTI-INFECTIVE AGENTS Achillion Pharmaceuticals, Inc. (US) 2012-02-08 EP claimed
WO-2010115184-A2 HYDROXYTHIENOQUINOLONES AND RELATED COMPOUNDS AS ANTI-INFECTIVE AGENTS ACHILLION PHARMACEUTICALS, INC. (US) 2010-10-07 WO claimed