SCHEMBL5373907

SCHEMBL5373907

Cc1ccc(Cc2ccc(=O)[nH]n2)c(F)c1Oc1cc(F)cc(C#N)c1

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.67
CYP2C9 P11712 1/20 0.67
CYP2C19 P33261 1/20 0.67
EPAS1 Q99814 11/20 0.38
THRA P10827 2/20 0.36
THRB P10828 2/20 0.36
KCNH2 Q12809 3/20 0.36
HAO1 Q9UJM8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373619 0.92 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19EPAS1THRA
SCHEMBL5364923 0.89 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19EPAS1THRA
SCHEMBL14559741 0.89 CYP3A4 (0.75) CYP3A4CYP2C9CYP2C19EPAS1THRA
SCHEMBL5365033 0.89 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19EPAS1THRA
SCHEMBL5366810 0.84 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5368884 0.83 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5668069 0.83 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19EPAS1KCNH2
SCHEMBL5373271 0.83 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19EPAS1THRA
SCHEMBL5377615 0.82 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19EPAS1THRA
SCHEMBL5377332 0.82 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19EPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed