SCHEMBL5377615

SCHEMBL5377615

CCc1ccc(Cc2ccc(=O)[nH]n2)c(F)c1Oc1cc(Cl)cc(C#N)c1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.60
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 1/20 0.56
KCNH2 Q12809 4/20 0.50
CYP2D6 P10635 1/20 0.35
THRA P10827 2/20 0.33
THRB P10828 2/20 0.33
SLC22A12 Q96S37 1/20 0.32
PGR P06401 1/20 0.32
VEGFA P15692 2/20 0.31
EPAS1 Q99814 2/20 0.31
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
P2RX3 P56373 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373843 0.91 CYP3A4 (0.65) CYP3A4CYP2C9CYP2C19KCNH2CYP2D6
SCHEMBL5382037 0.90 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19KCNH2CYP2D6
SCHEMBL5368884 0.86 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19KCNH2CYP2D6
SCHEMBL5373625 0.86 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL5373271 0.84 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL14559741 0.84 CYP3A4 (0.75) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL5385352 0.83 CYP3A4 (0.50) CYP3A4CYP2C9CYP2C19KCNH2SLC22A12
SCHEMBL4807889 0.83 CYP3A4 (0.84) CYP3A4CYP2C9CYP2C19KCNH2CYP2D6
SCHEMBL5365153 0.82 KCNH2 (0.46) CYP3A4CYP2C9CYP2C19KCNH2CYP2D6
SCHEMBL5373619 0.82 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19KCNH2THRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed