SCHEMBL5374835

SCHEMBL5374835

COc1ccc(-c2nc3cc(C)ccn3c2NCc2ccc3c(c2)OCO3)cc1OC

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 12/20 0.80
GAA P10253 11/20 0.80
ALDH1A1 P00352 10/20 0.80
RAB9A P51151 4/20 0.80
L3MBTL1 Q9Y468 4/20 0.80
MAPK1 P28482 4/20 0.80
NPSR1 Q6W5P4 3/20 0.80
KDM4E B2RXH2 8/20 0.74
HPGD P15428 5/20 0.74
SMN1; SMN2 Q16637 5/20 0.64
NPC1 O15118 2/20 0.64
TDP1 Q9NUW8 2/20 0.64
PKM P14618 1/20 0.64
TP53 P04637 2/20 0.64
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
TSHR P16473 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5370506 0.88 GAA (0.80) MAPTGAAALDH1A1RAB9AL3MBTL1
SCHEMBL2250301 0.87 GAA (0.68) MAPTGAAALDH1A1RAB9AL3MBTL1
SCHEMBL5372147 0.84 GAA (0.66) MAPTGAAALDH1A1RAB9AL3MBTL1
SCHEMBL5425036 0.83 NR1H4 (0.62) MAPTGAAALDH1A1RAB9AL3MBTL1
SCHEMBL5373182 0.76 NR1H4 (0.63) MAPTGAAALDH1A1RAB9AL3MBTL1
SCHEMBL2251270 0.76 GAA (0.68) MAPTGAAALDH1A1RAB9AL3MBTL1
SCHEMBL2253516 0.76 GAA (0.74) MAPTGAAALDH1A1RAB9AL3MBTL1
SCHEMBL2252724 0.75 GAA (0.75) MAPTGAAALDH1A1RAB9AL3MBTL1
SCHEMBL31344185 0.74 MAPT (0.79) MAPTGAAALDH1A1RAB9AL3MBTL1
SCHEMBL6285593 0.72 NR1H4 (0.48) MAPTGAAALDH1A1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007067711-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS FOR MODULATING TRPV1 AMPHORA DISCOVERY CORPORATION (US) 2007-06-14 WO disclosed