SCHEMBL5375820

SCHEMBL5375820

CCCC(CCC)S(=O)(=O)CC(N)C(=O)N(C(=O)OCc1ccccc1)[C@@H](Cc1cc(F)cc(F)c1)[C@H](O)CNCCC(C)C

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.49
CTSB P07858 14/20 0.49
CTSD P07339 2/20 0.40
ABCB1 P08183 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3352491 0.89 BACE1 (0.63) BACE1CTSBCTSD
SCHEMBL5375925 0.80 BACE1 (0.41) BACE1CTSBCTSDBACE2
SCHEMBL3350542 0.80 BACE1 (0.47) BACE1CTSBCTSD
SCHEMBL3351920 0.80 BACE1 (0.47) BACE1CTSBCTSD
SCHEMBL5388135 0.80 BACE1 (0.41) BACE1CTSBCTSD
SCHEMBL5383729 0.79 BACE1 (0.54) BACE1CTSBCTSD
SCHEMBL5377921 0.79 BACE1 (0.40) BACE1CTSBCTSDBACE2
SCHEMBL5369371 0.78 BACE1 (0.58) BACE1CTSBCTSD
SCHEMBL3357093 0.78 BACE1 (0.62) BACE1CTSBCTSD
SCHEMBL6700817 0.78 BACE1 (0.58) BACE1CTSBCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US disclosed