SCHEMBL5376006

SCHEMBL5376006

CCCCCCCc1nc(-c2ccncc2)cc(=O)[nH]1

nearest known ligand 0.90

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.90
GPR84 Q9NQS5 8/20 0.62
SMN1; SMN2 Q16637 1/20 0.52
XDH P47989 2/20 0.46
CDC7 O00311 1/20 0.44
DYRK3 O43781 1/20 0.44
ROCK2 O75116 1/20 0.44
MAP4K4 O95819 1/20 0.44
CDK1 P06493 1/20 0.44
CSF1R P07333 1/20 0.44
PIM1 P11309 1/20 0.44
PRKACA P17612 1/20 0.44
CDK2 P24941 1/20 0.44
MARK3 P27448 1/20 0.44
MAPK1 P28482 1/20 0.44
CSNK1A1 P48729 1/20 0.44
CSNK1D P48730 1/20 0.44
CLK2 P49760 1/20 0.44
GSK3A P49840 1/20 0.44
CDK7 P50613 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5381276 1.00 GSK3B (0.90) GSK3BGPR84SMN1; SMN2XDHCDC7
SCHEMBL5400097 1.00 GSK3B (0.90) GSK3BGPR84SMN1; SMN2XDHCDC7
SCHEMBL5381263 0.99 GSK3B (0.92) GSK3BGPR84SMN1; SMN2XDHCDC7
SCHEMBL5386254 0.94 GSK3B (1.00) GSK3BGPR84SMN1; SMN2XDHCDC7
SCHEMBL5380514 0.89 GSK3B (0.84) GSK3BGPR84SMN1; SMN2XDHCDC7
SCHEMBL3854866 0.83 SMN1; SMN2 (0.74) GSK3BGPR84SMN1; SMN2XDHCDC7
SCHEMBL5382475 0.82 GSK3B (0.77) GSK3BGPR84SMN1; SMN2XDH
SCHEMBL5387930 0.80 GSK3B (1.00) GSK3BGPR84SMN1; SMN2XDHCDC7
SCHEMBL5390457 0.79 GSK3B (0.72) GSK3BGPR84SMN1; SMN2XDHCDC7
SCHEMBL5381271 0.78 GSK3B (0.56) GSK3BGPR84CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO disclosed