SCHEMBL5376949

SCHEMBL5376949

N#Cc1ccc(Cl)cc1Oc1c(Cl)ccc(Cc2ccc(=O)[nH]n2)c1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
SLC22A12 Q96S37 2/20 0.35
SLC6A4 P31645 5/20 0.33
HTR2A P28223 3/20 0.33
KCNH2 Q12809 3/20 0.33
AKR1B1 P15121 2/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
PGGT1B P53609 1/20 0.33
CYP2D6 P10635 2/20 0.32
SLC6A2 P23975 2/20 0.32
NOS2 P35228 2/20 0.32
BCAT2 O15382 1/20 0.32
BCAT1 P54687 1/20 0.32
IDH1 O75874 2/20 0.32
EPHX2 P34913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367044 0.92 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19LMNAPOLB
SCHEMBL5364946 0.85 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19LMNAPOLB
SCHEMBL5364622 0.85 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19LMNAPOLB
SCHEMBL5373910 0.84 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19LMNAPOLB
SCHEMBL5368884 0.82 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19LMNAPOLB
SCHEMBL5373843 0.82 CYP3A4 (0.65) CYP3A4CYP2C9CYP2C19LMNAPOLB
SCHEMBL5370291 0.81 CYP3A4 (0.43) CYP3A4LMNAPOLBSLC22A12SLC6A4
SCHEMBL5368441 0.81 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19SLC6A4HTR2A
SCHEMBL5365045 0.80 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19SLC6A4HTR2A
SCHEMBL14559741 0.80 CYP3A4 (0.75) CYP3A4CYP2C9CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed