SCHEMBL5377008

SCHEMBL5377008

OC(c1ccccc1)(C(F)(F)F)C(F)(F)C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 14/20 0.53
NR1H3 Q13133 15/20 0.52
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
NR1I2 O75469 1/20 0.44
PTPN1 P18031 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9644838 0.93 NR1H3 (0.48) NR1H2NR1H3ALDH1A1TSHRNR1I2
SCHEMBL542694 0.87 NR1H3 (0.63) NR1H2NR1H3ALDH1A1TSHR
SCHEMBL2864482 0.87 NR1H3 (0.57) NR1H2NR1H3ALDH1A1TSHRPTPN1
Water SCHEMBL29107396 0.85 NR1H3 (0.61) NR1H2NR1H3ALDH1A1TSHR
SCHEMBL27702343 0.85 NR1H3 (0.61) NR1H2NR1H3ALDH1A1TSHR
SCHEMBL16886228 0.81 NR1H3 (0.57) NR1H2NR1H3ALDH1A1TSHR
SCHEMBL23149896 0.79 NR1H3 (0.50) NR1H2NR1H3ALDH1A1TSHRPTPN1
SCHEMBL26082774 0.79 NR1H3 (0.55) NR1H2NR1H3ALDH1A1TSHR
SCHEMBL3378017 0.78 TSHR (0.48) NR1H2NR1H3ALDH1A1TSHRPTPN1
SCHEMBL2228773 0.78 TSHR (0.48) NR1H2NR1H3ALDH1A1TSHRNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160449-B2 Proline chiral columns with broad chiral selectivity VANDERBILT UNIVERSITY (US) 2007-01-09 US disclosed
US-7141160-B2 Chiral columns with broad chiral selectivity V{dot over (a)}nderbilt University (US) 2006-11-28 US disclosed
US-20050092686-A1 Proline chiral columns with broad chiral selectivity LI, TINGYU 2005-05-05 US disclosed
EP-0302331-B1 ESTERS OF ARYLBISPERFLUORALKYLCARBINOLS, METHOD FOR THE PREPARATION OF THE SAME AND OF THE ARYLBISPERFLUORALKYLCARBINOLS IN QUESTION HOECHST AKTIENGESELLSCHAFT (DE) 1992-09-16 EP disclosed
US-5017719-A Esterification HOECHST AKTIENGESELLSCHAFT (DE) 1991-05-21 US disclosed
EP-0302331-A2 Esters of arylbisperfluoralkylcarbinols, method for the preparation of the same and of the arylbisperfluoralkylcarbinols in question HOECHST AKTIENGESELLSCHAFT (DE) 1989-02-08 EP disclosed