SCHEMBL2228773

SCHEMBL2228773

OC(c1ccccc1)(c1ccccc1)C(F)(F)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.48
ALDH1A1 P00352 2/20 0.48
PTPN1 P18031 1/20 0.43
NR1H2 P55055 6/20 0.41
NR1H3 Q13133 4/20 0.39
NR1I2 O75469 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP19A1 P11511 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA5A P35218 1/20 0.37
CA9 Q16790 1/20 0.37
HSD11B1 P28845 1/20 0.36
KCNN4 O15554 1/20 0.36
S1PR4 O95977 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5865852 0.84 TSHR (0.52) TSHRALDH1A1PTPN1NR1H2NR1H3
SCHEMBL3378017 0.80 TSHR (0.48) TSHRALDH1A1PTPN1NR1H2NR1H3
SCHEMBL9644838 0.80 NR1H3 (0.48) TSHRALDH1A1PTPN1NR1H2NR1H3
SCHEMBL5377008 0.78 NR1H2 (0.53) TSHRALDH1A1PTPN1NR1H2NR1H3
SCHEMBL7173455 0.78 CYP1A2 (0.48) TSHRALDH1A1PTPN1CYP1A2CYP2C9
SCHEMBL36629 0.78 CYP1A2 (0.48) TSHRALDH1A1PTPN1CYP1A2CYP2C9
SCHEMBL21135302 0.76 HSD11B1 (0.50) TSHRALDH1A1PTPN1NR1H2NR1H3
SCHEMBL7743285 0.75 CYP1A2 (0.46) TSHRALDH1A1PTPN1CYP1A2CYP2C9
SCHEMBL30915210 0.75 ALDH1A1 (0.70) TSHRALDH1A1PTPN1NR1H2CYP3A4
SCHEMBL7766770 0.75 ALDH1A1 (0.70) TSHRALDH1A1PTPN1NR1H2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10450253-B2 Preparation process of perfluoroalkyl compound with monohydroperfluoroalkane as starting material KANTO DENKA KOGYO CO., LTD. (JP) 2019-10-22 US disclosed
US-20190169107-A1 PREPARATION PROCESS OF PERFLUOROALKYL COMPOUND WITH MONOHYDROPERFLUOROALKANE AS STARTING MATERIAL NATIONAL UNIVERSITY CORPORATION GUNMA UNIVERSITY (JP) 2019-06-06 US disclosed
US-8084617-B2 Ionic liquids having fluoroalkyltrifluoroborate anions MERCK PATENT GMBH (DE) 2011-12-27 US disclosed
EP-2058319-B1 Use of perfluoralkylphosphines as perfluoroalkylation reagents MERCK PATENT GMBH (DE) 2011-08-17 EP disclosed
EP-1730157-B1 IONIC LIQUIDS COMPRISING FLUORALKYLTRIFFLUOROBORATE ANIONS MERCK PATENT GMBH (DE) 2011-07-27 EP disclosed
US-7632969-B2 Process for the preparation of perfluoroalkylphosphines and the use thereof as perfluoroalkylating reagents MERCK PATENT GMBH (DE) 2009-12-15 US disclosed
EP-2058319-A1 Method for manufacturing perfluoralkylphosphines and their application as perfluoralkylisation reagents Merck Patent GmbH (DE) 2009-05-13 EP disclosed
EP-1495037-B1 METHOD FOR THE PRODUCTION OF PERFLUOROALKYL PHOSPHINES AND THE USE THEREOF AS PERFLUOROALKYLATING REACTANTS MERCK PATENT GMBH (DE) 2009-02-25 EP disclosed
US-20070213538-A1 Ionic Liquids Having Fluoroalkyltrifluoroborate Anions MERCK PATENT GMBH (DE) 2007-09-13 US disclosed
US-20070191637-A1 Reacting a (perfluoroalkyl)phosphorane fluoride with a hydride ion donor such as triethylsilane, tripropylsilane or sodium borohydride while refluxing WELZ-BIERMANN URS 2007-08-16 US disclosed
US-7208626-B2 Method for the production of perfluoroalkyl phosphines and the use thereof as perfluoroalkylating reactants MERCK PATENT GESELLSCHAFT (DE) 2007-04-24 US disclosed
EP-1730157-A1 IONIC LIQUIDS COMPRISING FLUORALKYLTRIFFLUOROBORATE ANIONS MERCK PATENT GmbH (DE) 2006-12-13 EP disclosed
WO-2005105815-A1 IONIC LIQUIDS COMPRISING FLUORALKYLTRIFFLUOROBORATE ANIONS MERCK PATENT GMBH (DE) 2005-11-10 WO disclosed
US-20050131256-A1 Method for the production of perfluoroaldyl phosphines and the use thereof as perfluoroalkylating reactants MERCK PATENT GMBH (DE) 2005-06-16 US disclosed
US-20050119513-A1 Method for perfluoroalkylation by means of tris (perfluoroalkyl) phosphine oxides MERCK PATENT GMBH (DE) 2005-06-02 US disclosed
EP-1495037-A1 METHOD FOR THE PRODUCTION OF PERFLUOROALKYL PHOSPHINES AND THE USE THEREOF AS PERFLUOROALKYLATING REACTANTS MERCK PATENT GmbH (DE) 2005-01-12 EP disclosed
EP-1494982-A1 METHOD FOR PERFLUOROALKYLATION BY MEANS OF TRIS(PERFLUOROALKYL)PHOSPHINE OXIDES MERCK PATENT GmbH (DE) 2005-01-12 EP disclosed
WO-2003087020-A1 METHOD FOR PERFLUOROALKYLATION BY MEANS OF TRIS(PERFLUOROALKYL)PHOSPHINE OXIDES MERCK PATENT GMBH (DE) 2003-10-23 WO disclosed
WO-2003087113-A1 METHOD FOR THE PRODUCTION OF PERFLUOROALKYL PHOSPHINES AND THE USE THEREOF AS PERFLUOROALKYLATING REACTANTS MERCK PATENT GMBH (DE) 2003-10-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213538-A1 Ionic Liquids Having Fluoroalkyltrifluoroborate Anions AFF1, AFF2, AFF4 TSHR 2063/4885ALDH1A1 1258/4885PTPN1 1354/4885
US-20190169107-A1 PREPARATION PROCESS OF PERFLUOROALKYL COMPOUND WITH MONOHYDROPERFLUOROALKANE AS STARTING MATERIAL PFKFB1, PFKFB4, PFAS TSHR 2116/4885ALDH1A1 505/4885PTPN1 3911/4885
US-10450253-B2 Preparation process of perfluoroalkyl compound with monohydroperfluoroalkane as starting material PFKFB1, PFKFB4, PFAS TSHR 2116/4885ALDH1A1 505/4885PTPN1 3911/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.