SCHEMBL5377597

SCHEMBL5377597

C=Cc1cc(C#N)cc(Oc2c(Cl)ccc(Cc3ccc(=O)[nH]n3)c2F)c1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
KCNH2 Q12809 3/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368884 0.91 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL14570794 0.90 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL14559741 0.88 CYP3A4 (0.75) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL5373843 0.88 CYP3A4 (0.65) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL5373271 0.86 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL5331103 0.85 CYP3A4 (0.61) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL5373625 0.85 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL14570716 0.84 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL5368441 0.84 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19KCNH2THRA
SCHEMBL5364850 0.83 CYP3A4 (0.59) CYP3A4CYP2C9CYP2C19KCNH2THRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed