SCHEMBL5385352

SCHEMBL5385352

CCc1ccc(Cc2ccc(=O)[nH]n2)c(F)c1Oc1cc(C#N)ccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
KCNH2 Q12809 6/20 0.38
HTR2A P28223 3/20 0.38
SLC6A4 P31645 4/20 0.34
SLC6A3 Q01959 1/20 0.34
SLC22A12 Q96S37 1/20 0.33
S100A9 P06702 1/20 0.32
TRPV4 Q9HBA0 1/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
JAK3 P52333 1/20 0.32
PGR P06401 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
IDH1 O75874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5364946 0.93 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL5377555 0.92 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL5365393 0.90 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL5377646 0.87 CYP3A4 (0.67) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL5367044 0.87 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL5366810 0.83 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL5377615 0.83 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19KCNH2SLC22A12
SCHEMBL5368441 0.81 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL5374165 0.81 CYP3A4 (0.74) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL5373625 0.81 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19KCNH2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed