SCHEMBL5378548

SCHEMBL5378548

COc1ccc(CN2C[C@@H]3C(c4c(F)cc(N5CC(CO)OC5=O)cc4F)[C@@H]3C2)cc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CALML3 P27482 6/20 0.46
SIGMAR1 Q99720 9/20 0.44
GRM2 Q14416 2/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14370650 1.00 CALML3 (0.46) CALML3SIGMAR1GRM2MAOAMAOB
SCHEMBL5374997 0.86 F10 (0.44) CALML3GRM2MAOAMAOB
SCHEMBL14370645 0.86 F10 (0.44) CALML3GRM2MAOAMAOB
SCHEMBL14370651 0.86 GRM2 (0.41) SIGMAR1GRM2
SCHEMBL14370644 0.84 F10 (0.45) CALML3SIGMAR1MAOAMAOB
SCHEMBL5375233 0.83 MAOA (0.53) MAOAMAOB
SCHEMBL14370652 0.83 MAOA (0.53) MAOAMAOB
SCHEMBL14224728 0.78 MAOA (0.54) CALML3MAOAMAOB
SCHEMBL4881816 0.78 MAOA (0.54) CALML3MAOAMAOB
SCHEMBL5383280 0.77 MAOA (0.51) CALML3SIGMAR1GRM2MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7279494-B2 Antimicrobial [3.1.0] bicyclohexylphenyl-oxazolidinone derivatives and analogues PFIZER INC. (US) 2007-10-09 US disclosed
US-20050192325-A1 Antimicrobial [3.1.0] bicyclohexylphenyl-oxazolidinone derivatives and analogues RENSLO ADAM (US) 2005-09-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050192325-A1 Antimicrobial [3.1.0] bicyclohexylphenyl-oxazolidinone derivatives and analogues OXA1L, CYP51A1, CYP2C19 CALML3 3870/4885SIGMAR1 450/4885GRM2 3931/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.