SCHEMBL5379060

SCHEMBL5379060

Cc1nc2sc3c(c2c(-c2cccs2)c1CC=O)CCCC3

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.52
RAB9A P51151 4/20 0.52
ALDH1A1 P00352 4/20 0.52
HPGD P15428 3/20 0.52
MAPT P10636 3/20 0.52
KDM4E B2RXH2 3/20 0.52
TP53 P04637 2/20 0.52
HSD17B10 Q99714 2/20 0.52
CASP1 P29466 2/20 0.52
CASP7 P55210 2/20 0.52
LMNA P02545 2/20 0.52
HCRTR1 O43613 1/20 0.52
TSHR P16473 1/20 0.52
HTT P42858 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
NPC1 O15118 3/20 0.50
KMT2A Q03164 1/20 0.49
POLB P06746 1/20 0.42
CNR1 P21554 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319629 0.98 SMN1; SMN2 (0.51) SMN1; SMN2RAB9AALDH1A1HPGDMAPT
SCHEMBL132616 0.84 KMT2A (0.70) SMN1; SMN2RAB9AALDH1A1HPGDMAPT
SCHEMBL3476753 0.82 KMT2A (0.67) SMN1; SMN2RAB9AALDH1A1HPGDMAPT
SCHEMBL99721 0.80 KMT2A (0.53) SMN1; SMN2RAB9AALDH1A1HPGDMAPT
SCHEMBL15875975 0.79 KMT2A (0.52) SMN1; SMN2RAB9AALDH1A1HPGDMAPT
SCHEMBL4055394 0.79 HPGD (0.53) SMN1; SMN2RAB9AALDH1A1HPGDMAPT
SCHEMBL5319449 0.78 ALDH1A1 (0.50) SMN1; SMN2RAB9AALDH1A1HPGDMAPT
SCHEMBL4055923 0.78 SMN1; SMN2 (0.50) SMN1; SMN2RAB9AALDH1A1HPGDMAPT
SCHEMBL135414 0.77 KMT2A (0.48) KMT2A
SCHEMBL4059332 0.77 SMN1; SMN2 (0.53) SMN1; SMN2RAB9AALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828199-A1 THIENO-PYRIDINE DERIVATIVES AS GABA-B ALLOSTERIC ENHANCERS F. Hoffmann-Roche AG (CH) 2007-09-05 EP claimed
WO-2006063732-A1 THIENO-PYRIDINE DERIVATIVES AS GABA-B ALLOSTERIC ENHANCERS F.HOFFMANN-LA ROCHE AG (CH) 2006-06-22 WO claimed