SCHEMBL5380796

SCHEMBL5380796

CC1(c2cc(Cl)ccc2Cl)NC(=O)NC1=O

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 7/20 0.53
AKR1A1 P14550 2/20 0.53
PDE7A Q13946 1/20 0.41
HCAR2 Q8TDS4 1/20 0.40
PTGER3 P43115 1/20 0.40
LMNA P02545 1/20 0.40
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP8 P22894 1/20 0.39
MMP14 P50281 1/20 0.39
MMP17 Q9ULZ9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL542294 0.78 PTGER3 (0.41) AKR1B1AKR1A1PDE7APTGER3LMNA
SCHEMBL7099930 0.75 LMNA (0.51) AKR1B1AKR1A1LMNAMMP2MMP3
SCHEMBL542817 0.75 LMNA (0.51) AKR1B1AKR1A1LMNAMMP2MMP3
SCHEMBL542398 0.75 LMNA (0.55) AKR1B1LMNAMMP2
SCHEMBL25400175 0.73 LMNA (0.50) AKR1B1AKR1A1HCAR2LMNAMMP2
SCHEMBL29949390 0.73 LMNA (0.50) AKR1B1AKR1A1HCAR2LMNAMMP2
SCHEMBL29949272 0.71 LMNA (0.51) LMNAMMP2MMP14
SCHEMBL11001789 0.69 AKR1B1 (1.00) AKR1B1AKR1A1
SCHEMBL21940203 0.69 PDE7A (0.50) AKR1B1AKR1A1PDE7A
SCHEMBL8207892 0.69 TP53 (0.42) AKR1B1AKR1A1HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160449-B2 Proline chiral columns with broad chiral selectivity VANDERBILT UNIVERSITY (US) 2007-01-09 US disclosed
US-7160449-B2 Proline chiral columns with broad chiral selectivity VANDERBILT UNIVERSITY (US) 2007-01-09 US disclosed
US-7160449-B2 Proline chiral columns with broad chiral selectivity VANDERBILT UNIVERSITY (US) 2007-01-09 US disclosed
US-7141160-B2 Chiral columns with broad chiral selectivity V{dot over (a)}nderbilt University (US) 2006-11-28 US disclosed
US-20050092686-A1 Proline chiral columns with broad chiral selectivity LI, TINGYU 2005-05-05 US disclosed