SCHEMBL5391850

SCHEMBL5391850

CCOC(=O)C1CN(C2CC[N]2)C1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.45
ALDH1A1 P00352 8/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
NPC1 O15118 1/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14916903 0.78 MAPT (0.50) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL15495063 0.74 MAPT (0.49) MAPTALDH1A1MEN1KMT2A
SCHEMBL237380 0.72 MAPT (0.60) MAPTALDH1A1MEN1KMT2ACYP3A4
SCHEMBL8891623 0.72 MAPT (0.60) MAPTALDH1A1MEN1KMT2ACYP3A4
SCHEMBL2375356 0.72 MAPT (0.60) MAPTALDH1A1MEN1KMT2ACYP3A4
SCHEMBL4221 0.72
SCHEMBL7119330 0.72 TSHR (0.41) MAPTALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL233475 0.72 MAPT (0.51) MAPTALDH1A1MEN1KMT2ACYP3A4
Hydrochloric Acid SCHEMBL28788727 0.71
SCHEMBL23421852 0.71 ALDH1A1 (0.51) MAPTALDH1A1MEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007506696-A 2007-03-22 JP claimed
EP-1667980-A1 1,4-DISUBSTITUTED ISOQUINOLINE DERIVATIVES AS RAF-KINASE INHIBITORS USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES Novartis AG (CH) 2006-06-14 EP claimed
WO-2005028444-A1 1,4-DISUBSTITUTED ISOQUINILONE DERIVATIVES AS RAF-KINASE INHIBITORS USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES NOVARTIS AG (CH) 2005-03-31 WO claimed