SCHEMBL5400044

SCHEMBL5400044

Cc1nc(=O)cc(-c2cccnc2)[nH]1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.59
CYP19A1 P11511 2/20 0.56
KMT2A Q03164 1/20 0.52
PKN2 Q16513 1/20 0.48
PIK3C3 Q8NEB9 2/20 0.47
ALK Q9UM73 1/20 0.46
NPY5R Q15761 3/20 0.46
CYP3A4 P08684 2/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
BTK Q06187 1/20 0.44
CYP2E1 P05181 2/20 0.44
CYP2B6 P20813 2/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5382536 0.81 CYP19A1 (0.52) CYP2A6CYP19A1KMT2APKN2PIK3C3
SCHEMBL5377972 0.80 GSK3B (0.56) PKN2
SCHEMBL5384453 0.80 CYP19A1 (0.59) CYP19A1KMT2APKN2NPY5RALDH1A1
SCHEMBL5381418 0.79 CYP19A1 (0.54) CYP19A1KMT2APKN2PIK3C3NPY5R
SCHEMBL10840148 0.78 CYP19A1 (0.52) CYP2A6CYP19A1KMT2APKN2PIK3C3
SCHEMBL5400045 0.76 GSK3B (0.69) CYP2A6CYP19A1KMT2APIK3C3ALK
SCHEMBL5376057 0.76 KMT2A (0.54) CYP19A1KMT2ANPY5RALDH1A1BTK
SCHEMBL1606072 0.75 CYP19A1 (0.65) CYP2A6CYP19A1KMT2AALKNPY5R
SCHEMBL17518797 0.75 CYP2A6 (1.00) CYP2A6CYP19A1NPY5RCYP3A4ALDH1A1
SCHEMBL7946248 0.74 CYP19A1 (0.68) CYP2A6CYP19A1KMT2ANPY5RCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed