SCHEMBL5384453

SCHEMBL5384453

O=c1cc(-c2cccnc2)[nH]c(-c2ccccc2)n1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.59
HPGD P15428 2/20 0.54
NPY5R Q15761 2/20 0.53
KMT2A Q03164 1/20 0.51
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 2/20 0.49
GAA P10253 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
MAPT P10636 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
NPC1 O15118 1/20 0.49
STAT1 P42224 1/20 0.49
RAB9A P51151 1/20 0.49
KDM4C Q9H3R0 2/20 0.48
LDHA P00338 1/20 0.48
EPHX2 P34913 1/20 0.48
PKN2 Q16513 1/20 0.47
HPGDS O60760 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5381418 0.93 CYP19A1 (0.54) CYP19A1HPGDNPY5RKMT2AKDM4E
SCHEMBL5376057 0.87 KMT2A (0.54) CYP19A1HPGDNPY5RKMT2AKDM4E
SCHEMBL19665231 0.85 HPGD (0.53) HPGDNPY5RKMT2AKDM4EALDH1A1
SCHEMBL5381545 0.84 CDC7 (0.59) HPGDNPY5RKDM4EALDH1A1GAA
SCHEMBL31074829 0.81 SCN2A (0.47) CYP19A1HPGDNPY5RKMT2AKDM4E
SCHEMBL5400044 0.80 CYP2A6 (0.59) CYP19A1NPY5RKMT2AALDH1A1PKN2
SCHEMBL5385542 0.79 RAF1 (0.46) HPGDNPY5RKMT2AALDH1A1GAA
SCHEMBL5377577 0.77 CDC7 (0.49) HPGDNPY5RKDM4EALDH1A1MAPT
SCHEMBL5384455 0.77 GSK3B (0.75) CYP19A1HPGDNPY5RKMT2AKDM4E
SCHEMBL10840148 0.77 CYP19A1 (0.52) CYP19A1HPGDKMT2AALDH1A1PKN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO disclosed