SCHEMBL5407083

SCHEMBL5407083

CCn1c(Sc2cc(C#N)cc(C#N)c2)cnc1CNC(N)=O

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.33
ROCK2 O75116 1/20 0.32
KDR P35968 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
MTOR P42345 1/20 0.31
GSK3B P49841 1/20 0.31
PRKDC P78527 1/20 0.31
KCNH2 Q12809 1/20 0.31
ATM Q13315 1/20 0.31
ATR Q13535 1/20 0.31
JAK2 O60674 1/20 0.31
TYK2 P29597 1/20 0.31
JAK3 P52333 1/20 0.31
HSP90B1 P14625 1/20 0.31
PTGER4 P35408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4892053 0.80 IRAK4 (0.31) IRAK4
SCHEMBL4896675 0.67 TLR7 (0.31)
SCHEMBL4902450 0.64 HTR2C (0.32)
SCHEMBL4900565 0.64 HSP90B1 (0.30) HSP90B1
SCHEMBL4900191 0.64 HSP90B1 (0.32) HSP90B1
SCHEMBL6961868 0.63 F2 (0.31)
SCHEMBL6974137 0.63 CYP2C9 (0.32) HSP90B1
SCHEMBL4899905 0.62
SCHEMBL4902680 0.62 ALDH1A1 (0.35)
SCHEMBL4895868 0.62 AOC3 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740550-A1 SULPHUR-LINKED IMIDAZOLE COMPOUNDS FOR THE TREAMENT OF HIV Pfizer Limited (GB) 2007-01-10 EP disclosed
WO-2005100322-A1 SULPHUR-LINKED IMIDAZOLE COMPOUNDS FOR THE TREAMENT OF HIV PFIZER LIMITED (GB) 2005-10-27 WO disclosed