SCHEMBL5408472

SCHEMBL5408472

N#Cc1c(-c2cccs2)cc(-c2ccccc2)nc1OC(C(=O)O)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.57
ADORA1 P30542 3/20 0.57
ALDH1A1 P00352 8/20 0.47
HPGD P15428 8/20 0.47
KDM4E B2RXH2 7/20 0.47
GLA P06280 4/20 0.47
GAA P10253 3/20 0.47
CASP1 P29466 1/20 0.47
HSD17B10 Q99714 1/20 0.47
KMT2A Q03164 4/20 0.47
NPSR1 Q6W5P4 5/20 0.47
MEN1 O00255 3/20 0.47
PPARG P37231 3/20 0.47
NCOA2 Q15596 3/20 0.47
NCOA1 Q15788 3/20 0.47
SQOR Q9Y6N5 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
NCOA3 Q9Y6Q9 2/20 0.45
RXFP1 Q9HBX9 1/20 0.45
PIM1 P11309 4/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5414611 0.93 HPGD (0.54) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL5390378 0.92 ADORA2A (0.57) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL29442321 0.86 KDM4E (0.52) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL14385653 0.86 ALDH1A1 (0.53) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL29442296 0.86 KMT2A (0.48) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL22215932 0.86 KMT2A (0.48) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL14385234 0.86 ADORA2A (0.49) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL14385254 0.85 KMT2A (0.58) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL14385649 0.85 ADORA2A (0.46) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL14385269 0.84 KMT2A (0.49) ADORA2AADORA1ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007124545-A1 INTEGRASE INHIBITORS - 2 AVEXA LIMITED (AU) 2007-11-08 WO disclosed
WO-2007124545-A1 INTEGRASE INHIBITORS - 2 AVEXA LIMITED (AU) 2007-11-08 WO disclosed