SCHEMBL5409081

SCHEMBL5409081

Cc1ccc(S(=O)(=O)c2ccc(C(F)(F)F)cc2NC(=O)NC(Cc2ccc(NC(=O)c3c(Cl)cccc3Cl)cc2)C(=O)O)cc1

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.61
ITGA4 P13612 20/20 0.61
ITGA2 P17301 1/20 0.54
ITGB7 P26010 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5259894 1.00 ITGB1 (0.61) ITGB1ITGA4ITGA2ITGB7
SCHEMBL5405493 0.93 ITGB1 (0.51) ITGB1ITGA4ITGA2ITGB7
SCHEMBL5260018 0.93 ITGB1 (0.51) ITGB1ITGA4ITGA2ITGB7
SCHEMBL5388685 0.90 ITGB1 (0.61) ITGB1ITGA4ITGA2ITGB7
SCHEMBL5388690 0.85 ITGB1 (0.66) ITGB1ITGA4ITGA2ITGB7
SCHEMBL5261541 0.85 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7
SCHEMBL5261197 0.85 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7
SCHEMBL5261612 0.84 ITGB1 (0.64) ITGB1ITGA4ITGA2ITGB7
SCHEMBL5261619 0.84 ITGB1 (0.64) ITGB1ITGA4ITGA2ITGB7
SCHEMBL5258820 0.83 ITGB1 (0.58) ITGB1ITGA4ITGA2ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7253171-B2 Urea derivatives as integrin α4 antagonists LABORATORIOS ALMIRALL, S.A. (ES) 2007-08-07 US claimed
US-7253171-B2 Urea derivatives as integrin α4 antagonists LABORATORIOS ALMIRALL, S.A. (ES) 2007-08-07 US disclosed