SCHEMBL541099

SCHEMBL541099

O=COCc1ccc(C(F)(F)F)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.47
DAO P14920 1/20 0.45
MRGPRX4 Q96LA9 5/20 0.40
MGLL Q99685 2/20 0.37
SLC6A4 P31645 2/20 0.36
MAOB P27338 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.33
KMO O15229 1/20 0.33
NOTUM Q6P988 1/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5542683 0.88 IDO1 (0.39) IDO1DAOMRGPRX4MGLLSLC6A4
SCHEMBL18086871 0.85 IDO1 (0.44) IDO1DAOMRGPRX4MGLLSLC6A4
SCHEMBL5546553 0.82 KIF11 (0.45) IDO1DAO
SCHEMBL5722020 0.81 DAO (0.50) IDO1DAOMRGPRX4KMONOTUM
SCHEMBL95626 0.79 IDO1 (0.57) IDO1
SCHEMBL5536268 0.79 AR (0.45) IDO1SLC6A4AR
SCHEMBL5541400 0.78 IDO1 (0.49) IDO1MRGPRX4SLC6A4MAOBPTGDR2
SCHEMBL5547880 0.78 SCN3A (0.43) MRGPRX4PTGDR2KMO
SCHEMBL27810116 0.78 SLC6A4 (0.41) IDO1DAOMRGPRX4SLC6A4MAOB
SCHEMBL2091883 0.77 IDO1 (0.41) IDO1MAOBNOTUMAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414346-A1 AUTOTAXIN INHIBITORS Merck Patent GmbH (DE) 2012-02-08 EP disclosed
WO-2010112124-A1 AUTOTAXIN INHIBITORS MERCK PATENT GMBH (DE) 2010-10-07 WO disclosed