SCHEMBL5431933

SCHEMBL5431933

CCCN1C(=O)[C@@H]([C@H](O)C(C)C)NC(=O)C12CCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCN(Cc1c(C)nn(C3CCCCC3)c1C)CC2

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.48
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5343614 0.97 CCR5 (0.50) CCR5CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6641532 0.96 CCR5 (0.51) CCR5CYP2D6CYP2C9
SCHEMBL5345303 0.92 CCR5 (0.54) CCR5CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6010961 0.92 CCR5 (0.55) CCR5CYP2D6CYP2C9
SCHEMBL5344107 0.89 CCR5 (0.57) CCR5CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6010699 0.88 CCR5 (0.57) CCR5CYP2D6CYP2C9
SCHEMBL5347472 0.84 CCR5 (0.59) CCR5CYP2D6CYP2C9
SCHEMBL5348299 0.84 CCR5 (0.59) CCR5CYP2D6CYP2C9
SCHEMBL5346400 0.84 CCR5 (0.51) CCR5CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6010694 0.84 CCR5 (0.60) CCR5CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7262193-B2 Triazaspiro[5.5]undecane derivative and pharmaceutical composition comprising the same as active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2007-08-28 US claimed