SCHEMBL5437887

SCHEMBL5437887

O=C1Nc2cc(-c3ccco3)ccc2/C1=C\Nc1ccc(N2CCOCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 2/20 0.46
CSF1R P07333 1/20 0.45
RET P07949 2/20 0.41
MAPT P10636 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 3/20 0.40
LMNA P02545 1/20 0.40
APP P05067 1/20 0.40
POLB P06746 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
CASP1 P29466 1/20 0.40
SNCA P37840 1/20 0.40
BLM P54132 1/20 0.40
MCL1 Q07820 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CHEK1 O14757 4/20 0.40
TDP2 O95551 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5437889 1.00 PDGFRB (0.46) PDGFRBCSF1RRETMAPTMEN1
SCHEMBL5873816 1.00 PDGFRB (0.46) PDGFRBCSF1RRETMAPTMEN1
SCHEMBL7699129 0.88 CSF1R (0.40) PDGFRBCSF1RRETLMNATDP2
SCHEMBL7699131 0.88 CSF1R (0.40) PDGFRBCSF1RRETLMNATDP2
SCHEMBL5432746 0.83 RET (0.46) PDGFRBCSF1RRETCHEK1TDP2
SCHEMBL7703531 0.83 RET (0.46) PDGFRBCSF1RRETMAPTALDH1A1
SCHEMBL5432741 0.83 RET (0.46) PDGFRBCSF1RRETCHEK1TDP2
SCHEMBL7703527 0.83 RET (0.46) PDGFRBCSF1RRETMAPTALDH1A1
SCHEMBL5873980 0.83 RET (0.46) PDGFRBCSF1RRETCHEK1TDP2
SCHEMBL4996092 0.83 CHEK1 (0.51) PDGFRBCSF1RMAPTALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350747-B1 PROTEIN SERINE/THREONINE KINASE AND PROTEIN TYROSINE KINASE ENZYME INHIBITORS; ANGIOGENESIS INHIBITORS; ANTITUMOR AND ANTIPROLIFERATIVE AGENTS GLAXO WELLCOME INC. 2002-02-26 US claimed
EP-1165514-A1 3-(ANILINOMETHYLENE) OXINDOLES AS PROTEIN TYROSINE KINASE AND PROTEIN SERINE/THREONINE KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2002-01-02 EP claimed
WO-2000056710-A1 3-(ANILINOMETHYLENE) OXINDOLES AS PROTEIN TYROSINE KINASE AND PROTEIN SERINE/THREONINE KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2000-09-28 WO claimed
US-20070213403-A1 TAMOXIFEN RESPONSE IN PRE-AND POSTMENOPAUSAL BREAST CANCER PATIENTS FORSKARPATENT I SYD AB (SE) 2007-09-13 US disclosed