SCHEMBL5454042

SCHEMBL5454042

O=C(NCC1CCN(C(=O)OCc2ccc(F)cc2)CC1)c1cc[nH]c1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 4/20 0.61
TPSD1 Q9BZJ3 4/20 0.61
TPSG1 Q9NRR2 4/20 0.61
F2 P00734 2/20 0.61
PLG P00747 2/20 0.61
PRSS1 P07477 2/20 0.61
PRSS2 P07478 2/20 0.61
PRSS3 P35030 2/20 0.61
GRIN2B Q13224 12/20 0.57
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
KDM4E B2RXH2 1/20 0.44
PKM P14618 1/20 0.44
CYP3A4 P08684 1/20 0.43
F13A1 P00488 1/20 0.42
TGM2 P21980 1/20 0.42
TGM1 P22735 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367222 0.90 TPSAB1 (0.61) TPSAB1TPSD1TPSG1F2PLG
SCHEMBL5437286 0.90 TPSAB1 (0.61) TPSAB1TPSD1TPSG1F2PLG
SCHEMBL5448982 0.90 TPSAB1 (0.61) TPSAB1TPSD1TPSG1F2PLG
SCHEMBL5360257 0.90 TPSAB1 (0.60) TPSAB1TPSD1TPSG1F2PLG
SCHEMBL5362389 0.88 TPSAB1 (0.58) TPSAB1TPSD1TPSG1F2PLG
SCHEMBL5368080 0.87 GRIN2B (0.59) TPSAB1TPSD1TPSG1F2PLG
SCHEMBL5364146 0.86 TPSAB1 (0.61) TPSAB1TPSD1TPSG1F2PLG
SCHEMBL5367960 0.85 TPSAB1 (0.72) TPSAB1TPSD1TPSG1F2PLG
SCHEMBL5378288 0.84 TPSAB1 (0.66) TPSAB1TPSD1TPSG1F2PLG
SCHEMBL5358660 0.84 TPSAB1 (0.72) TPSAB1TPSD1TPSG1F2PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed