SCHEMBL5457783

SCHEMBL5457783

CCCCOP(=O)(OCCN)OCCCC

nearest known ligand 0.77

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.77
TSHR P16473 1/20 0.59
LPAR3 Q9UBY5 3/20 0.43
LPAR1 Q92633 2/20 0.43
LPAR2 Q9HBW0 2/20 0.43
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethylenediamine SCHEMBL31533530 0.95 CYP3A4 (0.85) CYP3A4TSHRLPAR3LPAR1LPAR2
SCHEMBL29212841 0.93 CYP3A4 (0.67) CYP3A4TSHRLPAR3LPAR1LPAR2
SCHEMBL28867253 0.91 CYP3A4 (0.64) CYP3A4TSHRLPAR3LPAR1LPAR2
SCHEMBL28867255 0.91 CYP3A4 (0.64) CYP3A4TSHRLPAR3LPAR1LPAR2
SCHEMBL31410773 0.91 CYP3A4 (0.64) CYP3A4TSHRLPAR3LPAR1LPAR2
SCHEMBL29212826 0.91 CYP3A4 (0.64) CYP3A4TSHRLPAR3LPAR1LPAR2
SCHEMBL28567051 0.91 CYP3A4 (0.77) CYP3A4TSHRLPAR3LPAR1LPAR2
SCHEMBL1020179 0.88 CYP3A4 (1.00) CYP3A4TSHRLPAR3LPAR1LPAR2
SCHEMBL27895927 0.88 CYP3A4 (1.00) CYP3A4TSHRLPAR3LPAR1LPAR2
SCHEMBL18570 0.88 CYP3A4 (1.00) CYP3A4TSHRLPAR3LPAR1LPAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7718688-B2 Nitrobenzindoles and their use in cancer therapy AUCKLAND UNISERVICES LIMITED (NZ) 2010-05-18 US disclosed
US-20080119442-A1 as hypoxia-selective drugs and radiosensitizers for cancer therapy; nitroreductase inhibitor; 1-(Chloromethyl)-5,6-dinitro-3-(5,6,7-trimethoxyindol-2-carbonyl)-1,2-dihydro-3H-benzo[e]indole; halogenation of naphthalene derivative followed by hydration and cyclization AUCKLAND UNISERVICES LIMITED (NZ) 2008-05-22 US disclosed
US-20070210476-A1 Machinable Resin Molded Product, Material For Forming The Same, And Model Made Of The Same SANYO CHEMICAL INDUSTRIES, LTD. (JP) 2007-09-13 US disclosed
EP-1728832-A1 MOLDING OF RESIN FOR CUTTING OPERATION, MATERIAL FOR FORMATION THEREOF AND MODEL Sanyo Chemical Industries, Ltd. (JP) 2006-12-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080119442-A1 as hypoxia-selective drugs and radiosensitizers for cancer therapy; nitroreductase inhibitor; 1-(Chloromethyl)-5,6-dinitro-3-(5,6,7-trimethoxyindol-2-carbonyl)-1,2-dihydro-3H-benzo[e]indole; halogenation of naphthalene derivative followed by hydration and cyclization HIF1AN, HYOU1, HIF1A CYP3A4 259/4885TSHR 1796/4885LPAR3 3437/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.