SCHEMBL545823

SCHEMBL545823

CCN1CCN(Cc2cccc(C(=O)NC(C)(C)C)c2)CC1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 3/20 0.50
HDAC1 Q13547 1/20 0.50
ACKR3 P25106 6/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
HIF1A Q16665 1/20 0.49
ALDH1A1 P00352 3/20 0.48
LMNA P02545 2/20 0.48
KDM4E B2RXH2 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
MAPT P10636 1/20 0.47
PTPN2 P17706 1/20 0.46
PKM P14618 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1017905 0.86 CHRM3 (0.61) CHRM3
Hydrochloric Acid SCHEMBL1018725 0.85 CHRM3 (0.60) CHRM3
SCHEMBL28052543 0.83 HDAC1 (0.45) CHRM3HDAC1ACKR3CYP2D6CYP2C9
SCHEMBL1020776 0.83 CYP2D6 (0.52) HDAC1ACKR3CYP2D6CYP2C9HIF1A
SCHEMBL1022120 0.83 GLS (0.49) CHRM3HDAC1ACKR3ALDH1A1LMNA
SCHEMBL12955045 0.82 CHRM3 (0.57) CHRM3CYP2D6CYP2C9HIF1ATDP1
SCHEMBL13701762 0.82 MAPT (0.49) CHRM3ALDH1A1LMNATDP1MAPT
SCHEMBL1017900 0.82 MEN1 (0.53) CHRM3ALDH1A1LMNAKDM4EMAPT
Hydrochloric Acid SCHEMBL1019737 0.81 CHRM3 (0.56) CHRM3CYP2D6CYP2C9HIF1A
SCHEMBL21319459 0.81 CYP2D6 (0.73) CYP2D6CYP2C9HIF1AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110687-B2 Bicyclic compounds with kinase inhibitory activity MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-07 US disclosed