SCHEMBL5471908

SCHEMBL5471908

NC(CS(=O)(=O)Cc1ccccc1OC(F)F)C(=O)NC1CCCCC1=O.O=C(O)C(CS(=O)(=O)Cc1ccccc1OC(F)F)NC(=O)N1CCOCC1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 14/20 0.41
CTSL P07711 10/20 0.41
CTSK P43235 6/20 0.41
CTSB P07858 7/20 0.36
TACR2 P21452 2/20 0.33
CTSH P09668 1/20 0.33
CTSC P53634 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14491116 0.92 CTSS (0.44) CTSSCTSLCTSKCTSB
SCHEMBL6842993 0.92 CTSS (0.44) CTSSCTSLCTSKCTSB
SCHEMBL6847855 0.89 CTSS (0.43) CTSSCTSLCTSKCTSBTACR2
SCHEMBL6847007 0.86 CTSS (0.43) CTSSCTSLCTSKCTSBTACR2
SCHEMBL5445303 0.85 KMT2A (0.35) POLB
SCHEMBL5436195 0.84 CTSS (0.46) CTSSCTSLCTSKCTSBCTSH
SCHEMBL6743322 0.84 CTSS (0.46) CTSSCTSLCTSKCTSBCTSH
SCHEMBL5445598 0.83 KMT2A (0.33) POLB
SCHEMBL5438734 0.80 KMT2A (0.34)
SCHEMBL1557679 0.75 CTSS (0.50) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7196099-B2 Compounds and compositions as cathepsin inhibitors AVENTIS PHARMACEUTICALS INC. (US) 2007-03-27 US disclosed