SCHEMBL5478945

SCHEMBL5478945

Cc1n[nH]c2ccc(-c3cc(N[C@@H](Cc4ccccc4)C(N)=O)cnc3-c3ccccc3O)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 17/20 0.51
FGFR1 P11362 16/20 0.51
FGFR3 P22607 16/20 0.51
AKT1 P31749 3/20 0.48
ROCK1 Q13464 3/20 0.48
ABL1 P00519 3/20 0.43
EGFR P00533 3/20 0.43
INSR P06213 3/20 0.43
RET P07949 3/20 0.43
SRC P12931 3/20 0.43
FGFR4 P22455 3/20 0.43
LTK P29376 3/20 0.43
KDR P35968 3/20 0.43
MERTK Q12866 3/20 0.43
ERBB4 Q15303 3/20 0.43
ALK Q9UM73 3/20 0.43
ERBB2 P04626 2/20 0.43
PDGFRB P09619 1/20 0.43
MAPK1 P28482 2/20 0.43
FLT1 P17948 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5475633 0.93 FGFR1 (0.49) FGFR2FGFR1FGFR3AKT1ROCK1
SCHEMBL5467170 0.87 AKT1 (0.48) FGFR2FGFR1FGFR3AKT1ABL1
SCHEMBL5467086 0.87 FGFR1 (0.52) FGFR2FGFR1FGFR3AKT1ROCK1
SCHEMBL4659680 0.85 CDK2 (0.54) FGFR2FGFR1FGFR3AKT1ROCK1
SCHEMBL4660832 0.84 AKT1 (0.55) FGFR2FGFR1FGFR3AKT1ROCK1
SCHEMBL4660844 0.84 AKT1 (0.55) FGFR2FGFR1FGFR3AKT1ROCK1
SCHEMBL28371016 0.81 FGFR2 (0.75) FGFR2FGFR1FGFR3ABL1EGFR
SCHEMBL4659759 0.78 CDK7 (0.57) FGFR2FGFR1FGFR3AKT1ROCK1
SCHEMBL4791250 0.78 AKT1 (0.77) AKT1ROCK1RETSRCMAPK1
SCHEMBL4791248 0.78 AKT1 (0.77) AKT1ROCK1RETSRCMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070185152-A1 Inhibitors of akt activity SMITHKLINE BEECHAM CORPORATION 2007-08-09 US claimed
US-20070185152-A1 Inhibitors of akt activity SMITHKLINE BEECHAM CORPORATION 2007-08-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070185152-A1 Inhibitors of akt activity AKT1, AKT1S1, AKT2 FGFR2 1337/4885FGFR1 1565/4885FGFR3 1449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.