SCHEMBL5480751

SCHEMBL5480751

[CH2]C(OC(C)=O)c1cccc(C(=O)C(C(=O)c2cccc(F)c2)=C2Nc3ccccc3N2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
ALDH1A1 P00352 4/20 0.36
LMNA P02545 3/20 0.36
GAA P10253 1/20 0.36
CYP3A4 P08684 4/20 0.34
GPR139 Q6DWJ6 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
USP2 O75604 2/20 0.33
CYP2D6 P10635 2/20 0.33
TSHR P16473 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
KCNK3 O14649 1/20 0.33
PARP1 P09874 1/20 0.33
POLB P06746 1/20 0.32
MAOB P27338 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2942138 0.85 CES2 (0.38) CES2CES1ALDH1A1LMNAGAA
SCHEMBL2948270 0.85 CES2 (0.38) CES2CES1ALDH1A1LMNAGAA
SCHEMBL4352918 0.84 CES2 (0.45) CES2CES1ALDH1A1LMNAGAA
SCHEMBL2942727 0.81 CES2 (0.34) CES2CES1ALDH1A1LMNAGAA
SCHEMBL2946482 0.80 CES2 (0.40) CES2CES1ALDH1A1LMNAGAA
SCHEMBL2942730 0.79 MEN1 (0.33) CES2CES1ALDH1A1LMNAGAA
SCHEMBL2946683 0.79 CES2 (0.38) CES2CES1ALDH1A1LMNAGAA
SCHEMBL2942146 0.78 CES2 (0.41) CES2CES1ALDH1A1LMNAGAA
SCHEMBL2943148 0.78 CES2 (0.43) CES2CES1ALDH1A1LMNAGAA
SCHEMBL2947177 0.78 CES2 (0.43) CES2CES1ALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1752452-A9 PROPANE-1,3-DIONE DERIVATIVE OR ITS SALT Astellas Pharma Inc. (JP) 2007-12-12 EP disclosed
EP-1752452-A1 PROPANE-1,3-DIONE DERIVATIVE OR ITS SALT Astellas Pharma Inc. (JP) 2007-02-14 EP disclosed