SCHEMBL5482649

SCHEMBL5482649

CCOC(=O)C(C)(C)Oc1ccc(CNC(=O)CCC#Cc2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 6/20 0.44
EPHX2 P34913 5/20 0.44
PPARG P37231 2/20 0.44
CYP3A4 P08684 2/20 0.44
ABCB11 O95342 1/20 0.44
CYP1A2 P05177 1/20 0.44
TSHR P16473 1/20 0.44
HTR2A P28223 1/20 0.44
PMP22 Q01453 1/20 0.44
NR1H4 Q96RI1 1/20 0.43
ACACB O00763 1/20 0.41
PPARD Q03181 1/20 0.41
HTT P42858 1/20 0.40
LMNA P02545 2/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
POLB P06746 1/20 0.39
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5483321 0.88 PPARA (0.50) PPARAEPHX2PPARGNR1H4ACACB
SCHEMBL5495786 0.86 POLB (0.49) PPARAEPHX2PPARGTSHRNR1H4
SCHEMBL5495781 0.85 EPHX2 (0.47) PPARAEPHX2PPARGNR1H4ACACB
SCHEMBL5486248 0.83 PPARA (0.44) PPARAEPHX2PPARGCYP3A4ABCB11
SCHEMBL8794052 0.76 PPARA (0.71) PPARAEPHX2PPARGCYP3A4ABCB11
SCHEMBL3873472 0.76 ACACB (0.45) EPHX2CYP3A4CYP1A2TSHRNR1H4
SCHEMBL4575602 0.74 PPARA (0.52) PPARAEPHX2PPARGCYP3A4ABCB11
SCHEMBL933617 0.74 EPHX2 (0.58) PPARAEPHX2PPARGCYP3A4NR1H4
SCHEMBL5486993 0.74 PPARA (0.42) PPARAPPARGCYP3A4ABCB11CYP1A2
SCHEMBL5489663 0.73 FBP1 (0.44) PPARAPPARGCYP3A4ABCB11CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7253192-B2 Phenyl derivatives comprising an acetylene group HOFFMANN-LA ROCHE INC. (US) 2007-08-07 US disclosed
US-20060004091-A1 Phenyl derivatives comprising an acetylene group F. HOFFMANN-LA ROCHE AG (CH) 2006-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004091-A1 Phenyl derivatives comprising an acetylene group PPARD, PPARA, PPARG PPARA 2/4885EPHX2 1651/4885PPARG 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.