SCHEMBL5482684

SCHEMBL5482684

NCCCn1nc2c(c1C(=O)O)CCc1cc(O)c(CCC(F)(F)F)cc1-2

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.31
CDK2 P24941 1/20 0.31
OPRD1 P41143 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1655959 0.97 OPRD1 (0.34) PDPK1CDK2OPRD1
Trifluoroacetic Acid SCHEMBL6788050 0.88 OPRD1 (0.32) PDPK1CDK2OPRD1
SCHEMBL1655960 0.86 PLK1 (0.31) PDPK1CDK2
Trifluoroacetic Acid SCHEMBL4267112 0.84 KDM1A (0.33) PDPK1CDK2OPRD1RORC
Trifluoroacetic Acid SCHEMBL6793385 0.84 S1PR1 (0.32) PDPK1CDK2OPRD1RORC
Trifluoroacetic Acid SCHEMBL6787805 0.83 CDK2 (0.36) PDPK1CDK2OPRD1RORC
SCHEMBL6792318 0.82 PDPK1 (0.35) PDPK1CDK2
SCHEMBL6792438 0.81 PDPK1 (0.34) PDPK1CDK2
Bromide SCHEMBL1655616 0.81 PDPK1 (0.34) PDPK1CDK2
Trifluoroacetic Acid SCHEMBL6791782 0.80 PDPK1 (0.33) PDPK1CDK2OPRD1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824498-A2 METHODS AND COMPOSITIONS FOR TREATING CELLULAR PROLIFERATIVE DISEASES THE MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2007-08-29 EP disclosed
WO-2006053315-A2 METHODS AND COMPOSITIONS FOR TREATING CELLULAR PROLIFERATIVE DISEASES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2006-05-18 WO disclosed