SCHEMBL5484456

SCHEMBL5484456

COc1ccc(N2CCCCC2)c(N)c1.COc1ccc(N2CCCCC2)c(Nc2cc(C(F)(F)F)nc(-c3cccnc3)n2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
HSD17B10 Q99714 3/20 0.44
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2C19 P33261 3/20 0.44
CYP2C9 P11712 2/20 0.44
ALOX15 P16050 2/20 0.44
TSHR P16473 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
GALR2 O43603 6/20 0.39
ABCG2 Q9UNQ0 2/20 0.39
GALR1 P47211 3/20 0.38
HDAC1 Q13547 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP2D6 P10635 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5484543 0.95 HSD17B10 (0.48) KDM4EHSD17B10CYP1A2CYP3A4CYP2C19
SCHEMBL5482995 0.80 TSHR (0.48) KDM4EHSD17B10CYP1A2CYP3A4CYP2C19
SCHEMBL5486944 0.80 CYP11B2 (0.44) KDM4EHSD17B10CYP1A2CYP3A4CYP2C19
SCHEMBL5477008 0.80 ABL1 (0.47) KDM4EHSD17B10CYP1A2CYP3A4CYP2C19
SCHEMBL5489633 0.79 CYP11B2 (0.44) KDM4EHSD17B10CYP1A2CYP3A4CYP2C19
SCHEMBL5484057 0.75 ABCG2 (0.54) KDM4EHSD17B10CYP1A2CYP3A4CYP2C19
SCHEMBL5484062 0.74 ABCG2 (0.59) CYP1A2CYP3A4CYP2C19CYP2C9TSHR
SCHEMBL14493019 0.73 ABCG2 (0.47) KDM4EHSD17B10CYP1A2CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL5482581 0.72 ABCG2 (0.47) KDM4EHSD17B10CYP1A2CYP3A4CYP2C19
SCHEMBL5485895 0.72 KMT2A (0.45) KDM4EHSD17B10CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7226927-B2 Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators of caspases and inducers of apoptosis and the use thereof CYTOVIA, INC. (US) 2007-06-05 US disclosed