SCHEMBL5485326

SCHEMBL5485326

CCCCc1cc(C(F)(F)F)c([N+](=O)[O-])cc1OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
POLB P06746 1/20 0.39
PTGES O14684 1/20 0.39
CTSV O60911 2/20 0.39
CTSL P07711 2/20 0.39
NR1H4 Q96RI1 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.38
MTNR1A P48039 1/20 0.38
CYP19A1 P11511 3/20 0.38
PTGER1 P34995 1/20 0.38
PTGER4 P35408 1/20 0.38
PTGER3 P43115 1/20 0.38
PTGER2 P43116 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
HTR1A P08908 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5052984 0.81 HTR2A (0.43) ALDH1A1MAPT
SCHEMBL394870 0.81 MEN1 (0.47) MEN1KMT2AMAPTPOLBPTGES
SCHEMBL21629482 0.78 MEN1 (0.45) MEN1KMT2AMAPTPOLBPTGES
SCHEMBL2970281 0.76 PTGES (0.55) MEN1KMT2AMAPTPOLBPTGES
SCHEMBL2570775 0.74 POLB (0.43) MEN1KMT2AMAPTPOLBPTGES
SCHEMBL27592053 0.73 MEN1 (0.46) MEN1KMT2AMAPTPOLBPTGES
SCHEMBL2013356 0.73 POLB (0.43) MEN1KMT2AMAPTPOLBPTGES
SCHEMBL8808389 0.73 PTGES (0.51) MEN1KMT2AMAPTPOLBPTGES
SCHEMBL11738169 0.72 MEN1 (0.43) MEN1KMT2AALDH1A1MAPTPOLB
SCHEMBL8316270 0.72 MEN1 (0.55) MEN1KMT2AALDH1A1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed