SCHEMBL5485843

SCHEMBL5485843

CNCCN(C)c1cccc2[nH]c(C(C)NC3CCCc4cccnc43)nc12

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 16/20 0.42
PARP1 P09874 2/20 0.36
CYP2D6 P10635 2/20 0.34
CHRM2 P08172 1/20 0.34
DRD2 P14416 1/20 0.34
OPRM1 P35372 1/20 0.34
KCNH2 Q12809 1/20 0.34
SLC40A1 Q9NP59 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4879547 0.78 CXCR4 (0.57) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL5485849 0.78 CXCR4 (0.43) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL4884724 0.69 CXCR4 (0.43) CXCR4CYP2D6CHRM2KCNH2
SCHEMBL4882916 0.68 CXCR4 (0.57) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL4882672 0.68 HDAC1 (0.48) CXCR4CYP2D6
SCHEMBL4113740 0.68 HDAC1 (0.48) CXCR4CYP2D6
SCHEMBL20848115 0.67 GAA (0.47) CXCR4CYP2D6KCNH2
SCHEMBL13069026 0.67 GAA (0.47) CXCR4CYP2D6KCNH2
SCHEMBL2510199 0.65 CXCR4 (0.43) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL2084443 0.64 CXCR4 (0.50) CXCR4CYP2D6CHRM2DRD2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1789045-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-30 EP disclosed
WO-2006023400-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-03-02 WO disclosed