SCHEMBL4884724

SCHEMBL4884724

CN1CCN(c2cccc3[nH]c([C@H](CO)NC4CCCc5cccnc54)nc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 17/20 0.43
HTR6 P50406 3/20 0.40
CYP2D6 P10635 3/20 0.40
ACE P12821 1/20 0.39
KCNH2 Q12809 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CYP3A4 P08684 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4889224 0.81 CXCR4 (0.51) CXCR4CYP2D6ACEKCNH2CHRM2
SCHEMBL4878573 0.81 HTR6 (0.51) CXCR4HTR6CYP2D6KCNH2CHRM2
SCHEMBL4878647 0.79 CXCR4 (0.44) CXCR4HTR6CYP2D6ACEKCNH2
SCHEMBL4889721 0.79 HTR6 (0.50) CXCR4HTR6CYP2D6KCNH2
SCHEMBL4886975 0.77 CXCR4 (0.52) CXCR4CYP2D6KCNH2CHRM2CHRM4
SCHEMBL4889158 0.76 HTR6 (0.53) CXCR4HTR6CYP2D6KCNH2
SCHEMBL4885967 0.75 CXCR4 (0.44) CXCR4ACEKCNH2CHRM2CHRM4
SCHEMBL4887285 0.74 CXCR4 (0.56) CXCR4CYP2D6KCNH2CHRM2CYP3A4
SCHEMBL4889717 0.73 CXCR4 (0.60) CXCR4KCNH2
SCHEMBL4881658 0.73 CXCR4 (0.60) CXCR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080045537-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2008-02-21 US disclosed
US-20080045537-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2008-02-21 US disclosed
US-20080045537-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2008-02-21 US disclosed
EP-1789045-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-30 EP disclosed
WO-2006023400-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-03-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045537-A1 Chemical Compounds CCR5, CXCR4, CXCR3 CXCR4 2/4885HTR6 2334/4885CYP2D6 4070/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.