SCHEMBL5486124

SCHEMBL5486124

N#Cc1cccc(C(=O)c2sc(Nc3ccc([N+]4(C5CCNCC5)CCCC(O)C4)cc3)nc2N)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 10/20 0.47
CDK2 P24941 10/20 0.47
ZAP70 P43403 1/20 0.45
GSK3A P49840 2/20 0.45
GSK3B P49841 2/20 0.45
CDK5 Q00535 8/20 0.44
CDK5R1 Q15078 8/20 0.44
CDK4 P11802 1/20 0.41
CCND1 P24385 1/20 0.41
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
MAPK14 Q16539 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5495558 0.92 CCNA2 (0.50) CCNA2CDK2ZAP70GSK3AGSK3B
SCHEMBL5487553 0.91 GSK3A (0.56) CCNA2CDK2ZAP70GSK3AGSK3B
SCHEMBL5488900 0.90 CDK5 (0.57) CCNA2CDK2ZAP70CDK5CDK5R1
SCHEMBL5483582 0.87 CCNA2 (0.58) CCNA2CDK2ZAP70CDK5CDK5R1
SCHEMBL5488707 0.86 TUBB8B (0.43) CCNA2CDK2GSK3AGSK3BCDK5
SCHEMBL5483911 0.86 CDK5 (0.44) CCNA2CDK2CDK5CDK5R1NPC1
SCHEMBL5484920 0.86 CDK5 (0.47) CCNA2CDK2GSK3AGSK3BCDK5
SCHEMBL5485272 0.86 CCNA2 (0.47) CCNA2CDK2GSK3AGSK3BCDK5
SCHEMBL5479292 0.86 NPC1 (0.47) CCNA2CDK2GSK3AGSK3BCDK5
SCHEMBL5481882 0.85 NPC1 (0.54) CCNA2CDK2GSK3AGSK3BCDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740576-A1 NOVEL PIPERIDINE SUBSTITUTED DIAMINOTHIAZOLES F. Hoffman-la Roche AG (CH) 2007-01-10 EP disclosed
WO-2005103034-A1 NOVEL PIPERIDINE SUBSTITUTED DIAMINOTHIAZOLES F. HOFFMAN-LA ROCHE AG (CH) 2005-11-03 WO disclosed