Bicarbonate

Bicarbonate

SCHEMBL5487332

COC(=O)c1ccc(C(C)(C)C)cc1OCC(F)(F)F.O=C([O-])[O-].[K+].[K+]

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
ALDH1A1 P00352 2/20 0.44
EGFR P00533 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.41
SCN8A Q9UQD0 4/20 0.40
SCN10A Q9Y5Y9 4/20 0.40
FFAR4 Q5NUL3 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
UGCG Q16739 2/20 0.39
NR1H4 Q96RI1 1/20 0.39
POLB P06746 1/20 0.39
RAB9A P51151 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2008247 0.95 CFTR (0.50) CFTRCYP1A2CYP2C9ALDH1A1EGFR
SCHEMBL2008596 0.82 RAB9A (0.44) CYP1A2CYP2C9ALDH1A1KDM4EMRGPRX4
SCHEMBL1547094 0.80 TDP1 (0.59) CFTRCYP1A2CYP2C9ALDH1A1EGFR
SCHEMBL2006511 0.79 EGFR (0.46) CFTRALDH1A1EGFRKDM4EFFAR4
SCHEMBL25247535 0.79 FFAR4 (0.56) CFTRCYP1A2CYP2C9ALDH1A1KDM4E
SCHEMBL20505135 0.78 CYP1A2 (0.50) CFTRCYP1A2CYP2C9ALDH1A1KDM4E
SCHEMBL12244969 0.76 MAPT (0.56) CFTRALDH1A1EGFRKDM4ENR1H4
SCHEMBL3784216 0.74 KDM4E (0.46) CFTRCYP1A2CYP2C9ALDH1A1KDM4E
SCHEMBL3152664 0.74 EGFR (0.40) CFTRALDH1A1EGFRKDM4ETDP1
SCHEMBL17708165 0.74 CFTR (0.56) CFTRALDH1A1EGFRKDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1753727-A1 NOVEL CIS-IMIDAZOLINES F.HOFFMANN-LA ROCHE AG (CH) 2007-02-21 EP disclosed
WO-2005110996-A1 NOVEL CIS-IMIDAZOLINES F.HOFFMANN-LA ROCHE AG (CH) 2005-11-24 WO disclosed