SCHEMBL5493875

SCHEMBL5493875

Cc1cc(Nc2ncnc3cccc(OC[C@H](C)CC(N)=O)c23)ccc1OCc1cscn1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 19/20 0.53
EGFR P00533 7/20 0.50
KCNH2 Q12809 6/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4481289 0.85 ERBB2 (0.56) ERBB2EGFRKCNH2
SCHEMBL4480709 0.84 ERBB2 (0.67) ERBB2EGFRKCNH2
SCHEMBL5490957 0.82 EGFR (0.55) ERBB2EGFRKCNH2
SCHEMBL4483658 0.81 ERBB2 (0.53) ERBB2EGFRKCNH2
SCHEMBL5699203 0.81 EGFR (0.54) ERBB2EGFRKCNH2
SCHEMBL4483967 0.81 ERBB2 (0.55) ERBB2EGFRKCNH2
SCHEMBL4472955 0.81 EGFR (0.51) ERBB2EGFRKCNH2
SCHEMBL4473685 0.80 ERBB2 (0.52) ERBB2EGFRKCNH2
SCHEMBL3807571 0.80 EGFR (0.54) ERBB2EGFRKCNH2
SCHEMBL3816930 0.79 ERBB2 (0.62) ERBB2EGFRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007511491-A 2007-05-10 JP claimed
EP-1685116-A1 QUINAZOLINE DERIVATIVES AstraZeneca AB (SE) 2006-08-02 EP claimed
WO-2005051923-A1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2005-06-09 WO claimed