SCHEMBL5494843

SCHEMBL5494843

CC(C)(C)OC(=O)C1CCc2ccccc2N1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
MTNR1A P48039 4/20 0.44
EPHX2 P34913 1/20 0.44
MAPK1 P28482 1/20 0.41
HTR1A P08908 4/20 0.39
HTR2A P28223 4/20 0.39
DRD3 P35462 4/20 0.39
MASP2 O00187 1/20 0.39
F2 P00734 1/20 0.39
DRD2 P14416 4/20 0.37
HTR2C P28335 2/20 0.37
MTNR1B P49286 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17647218 0.92 MAPT (0.47) SMYD3GAAMAPTMTNR1AEPHX2
SCHEMBL27358248 0.87 GAA (0.61) SMYD3GAAMAPTMTNR1AEPHX2
SCHEMBL7294748 0.87 GAA (0.61) SMYD3GAAMAPTMTNR1AEPHX2
SCHEMBL6847865 0.84 SMYD3 (0.39) SMYD3GAAMAPTMTNR1AEPHX2
SCHEMBL926907 0.84 SMYD3 (0.56) SMYD3GAAMAPTMTNR1AHTR1A
SCHEMBL30357995 0.84 SMYD3 (0.56) SMYD3GAAMAPTMTNR1AHTR1A
SCHEMBL8567081 0.84 SMYD3 (0.56) SMYD3GAAMAPTMTNR1AHTR1A
SCHEMBL7433964 0.84 SMYD3 (0.56) SMYD3GAAMAPTMTNR1AHTR1A
Oxalic Acid SCHEMBL7294772 0.83 MAPT (0.60) SMYD3GAAMAPTMTNR1AEPHX2
Hydrochloric Acid SCHEMBL5424922 0.82 SMYD3 (0.54) SMYD3GAAMAPTMTNR1AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed
EP-1399445-A2 SUBSTITUTED PYRROLOQUINOLINES AND PYRIDOQUINOLINES AS SEROTONIN AGONISTS AND ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-03-24 EP disclosed
WO-2002059124-A2 SUBSTITUTED PYRROLOQUINOLINES AND PYRIDOQUINOLINES AS SEROTONIN AGONISTS AND ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2002-08-01 WO disclosed
EP-1114035-A1 QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL APPLICATIONS THEREOF SUNTORY LIMITED (JP) 2001-07-11 EP disclosed
WO-2000010982-A1 QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL APPLICATIONS THEROF SUNTORY LIMITED (JP) 2000-03-02 WO disclosed
CN-1140174-A Piperidine derivatives, process for preparation thereof and application thereof in therapeutics SYNTHELABO (FR) 1997-01-15 CN disclosed