SCHEMBL5497263

SCHEMBL5497263

c1ccc(-c2cc3ccncc3nc2-c2ccc(CN3CCC(c4n[nH]c(-c5ccccn5)n4)CC3)cc2)cc1

nearest known ligand 0.75

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 19/20 0.75
AKT2 P31751 19/20 0.75
KCNH2 Q12809 4/20 0.54
AKT3 Q9Y243 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5499246 0.94 AKT1 (0.75) AKT1AKT2KCNH2AKT3
SCHEMBL2356455 0.86 AKT1 (0.62) AKT1AKT2KCNH2
SCHEMBL1137849 0.86 AKT1 (0.59) AKT1AKT2KCNH2AKT3
SCHEMBL12410248 0.85 AKT1 (0.60) AKT1AKT2KCNH2
SCHEMBL2271522 0.85 AKT1 (0.58) AKT1AKT2KCNH2AKT3
SCHEMBL1059047 0.84 KCNH2 (0.76) AKT1AKT2KCNH2
SCHEMBL1138090 0.84 AKT1 (0.54) AKT1AKT2KCNH2AKT3
Hydrochloric Acid SCHEMBL1501644 0.83 KCNH2 (0.75) AKT1AKT2KCNH2
SCHEMBL1501777 0.83 AKT1 (0.58) AKT1AKT2KCNH2
SCHEMBL2281065 0.83 AKT1 (0.56) AKT1AKT2KCNH2AKT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1827436-A2 INHIBITORS OF AKT ACTIVITY Merck & Co., Inc. (US) 2007-09-05 EP claimed
WO-2006065601-A2 INHIBITORS OF AKT ACTIVITY MERCK & CO., INC. (US) 2006-06-22 WO claimed