SCHEMBL5497501

SCHEMBL5497501

CCC(NC(c1ccccc1)(c1ccccc1)c1ccccc1)C(O)CC(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 2/20 0.44
KIF11 P52732 1/20 0.39
GRIN1 Q05586 4/20 0.37
GRIN2A Q12879 4/20 0.37
GRIN2D O15399 3/20 0.37
GRIN2C Q14957 3/20 0.37
GRIN2B Q13224 2/20 0.37
TRPA1 O75762 2/20 0.37
LMNA P02545 1/20 0.34
PSMB8 P28062 1/20 0.33
PSMB5 P28074 1/20 0.33
CACNA1F O60840 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
ADRA2B P18089 1/20 0.33
CHRM3 P20309 1/20 0.33
ADRA1A P35348 1/20 0.33
HRH1 P35367 1/20 0.33
OPRK1 P41145 1/20 0.33
CACNA1D Q01668 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3862734 0.87 KCNN4 (0.50) KCNN4KIF11GRIN1GRIN2AGRIN2D
SCHEMBL3862881 0.87 KCNN4 (0.50) KCNN4KIF11GRIN1GRIN2AGRIN2D
SCHEMBL3666885 0.83 KCNN4 (0.50) KCNN4KIF11GRIN1GRIN2AGRIN2D
SCHEMBL4484584 0.83 KCNN4 (0.50) KCNN4KIF11GRIN1GRIN2AGRIN2D
SCHEMBL3307096 0.83 KCNN4 (0.50) KCNN4KIF11GRIN1GRIN2AGRIN2D
SCHEMBL3853261 0.83 KCNN4 (0.50) KCNN4KIF11GRIN1GRIN2AGRIN2D
SCHEMBL6565005 0.81 KCNN4 (0.47) KCNN4KIF11GRIN1GRIN2AGRIN2D
SCHEMBL3852207 0.81 KCNN4 (0.47) KCNN4KIF11GRIN1GRIN2AGRIN2D
SCHEMBL3854524 0.81 KCNN4 (0.47) KCNN4KIF11GRIN1GRIN2AGRIN2D
SCHEMBL3853041 0.78 KCNN4 (0.47) KCNN4KIF11GRIN1GRIN2AGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1529047-B1 NEW PURINE DERIVATIVES CYCLACEL LTD (GB) 2007-02-21 EP disclosed