SCHEMBL5497573

SCHEMBL5497573

CCC(CC1CC1)Nc1nc(C)nc2c1CCN2c1ccc(C(F)(F)F)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 10/20 0.41
SCN9A Q15858 2/20 0.34
PHGDH O43175 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5493014 0.91 CRHR1 (0.51) CRHR1PHGDHCYP1A2CYP2C19
SCHEMBL5492052 0.79 CRHR1 (0.50) CRHR1
SCHEMBL5497565 0.78 CRHR1 (0.38) CRHR1SCN9APHGDHCYP1A2CYP2C19
SCHEMBL5495331 0.78 CRHR1 (0.50) CRHR1
SCHEMBL5496957 0.78 CRHR1 (0.43) CRHR1SCN9APHGDHCYP1A2CYP2C19
SCHEMBL6746234 0.77 CRHR1 (0.57) CRHR1PHGDHCYP1A2CYP2C19
SCHEMBL5497563 0.76 CRHR1 (0.46) CRHR1CYP2C19
SCHEMBL5497559 0.75 CRHR1 (0.40) CRHR1SCN9APHGDHCYP1A2CYP2C19
SCHEMBL5489958 0.73 CRHR1 (0.55) CRHR1PHGDH
SCHEMBL5489901 0.73 CRHR1 (0.41) CRHR1SCN9APHGDHCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7279474-B2 Substituted pyrrolo[2,3-d]pyrimidines as antagonists of the corticotropin releasing factor (CRF) GLAXO GROUP LIMITED (GB) 2007-10-09 US disclosed