SCHEMBL5499490

SCHEMBL5499490

CC(=O)Nc1ccc(-c2nc(C(S)c3cccc(CCC(=O)NN4CCN(C)CC4)n3)nc(N)c2C#N)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.47
ADORA2A P29274 3/20 0.47
IKBKB O14920 6/20 0.37
ADORA3 P0DMS8 2/20 0.37
ADORA2B P29275 1/20 0.37
CHUK O15111 2/20 0.34
MAP4K4 O95819 2/20 0.34
MAPK8 P45983 2/20 0.34
ITK Q08881 2/20 0.34
CLK4 Q9HAZ1 2/20 0.34
PRKD3 O94806 1/20 0.34
CDK2 P24941 1/20 0.34
MAPK9 P45984 1/20 0.34
CLK2 P49760 1/20 0.34
MAPK10 P53779 1/20 0.34
MAP4K2 Q12851 1/20 0.34
PASK Q96RG2 1/20 0.34
SRPK1 Q96SB4 1/20 0.34
MAP4K5 Q9Y4K4 1/20 0.34
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL946096 0.99 ADORA1 (0.47) ADORA1ADORA2AIKBKBADORA3ADORA2B
SCHEMBL27663322 0.90 ADORA1 (0.58) ADORA1ADORA2AIKBKBADORA3ADORA2B
SCHEMBL27663397 0.87 ADORA1 (0.53) ADORA1ADORA2AIKBKBADORA3CHUK
SCHEMBL950112 0.87 ADORA1 (0.46) ADORA1ADORA2AIKBKBADORA3ADORA2B
Hydrochloric Acid SCHEMBL945957 0.85 ADORA1 (0.45) ADORA1ADORA2AIKBKBADORA3ADORA2B
SCHEMBL3737757 0.85 ADORA1 (0.45) ADORA1ADORA2AIKBKBADORA3ADORA2B
SCHEMBL945816 0.85 ADORA1 (0.45) ADORA1ADORA2AIKBKBADORA3ADORA2B
SCHEMBL28761086 0.85 ADORA1 (0.52) ADORA1ADORA2AIKBKBADORA3CHUK
SCHEMBL27663484 0.85 ADORA1 (0.46) ADORA1ADORA2AIKBKBADORA3ADORA2B
Hydrochloric Acid SCHEMBL3740316 0.84 ADORA1 (0.44) ADORA1ADORA2AIKBKBADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740574-B1 4-AMINO-5-CYANOPYRIMIDINE DERIVATIVES OTSUKA PHARMA CO LTD (JP) 2007-06-27 EP disclosed