SCHEMBL5499583

SCHEMBL5499583

O=S(=O)(Cc1ccccc1)N(CCCSc1nc2ccccc2[nH]1)C1CC1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.55
ALDH1A1 P00352 3/20 0.54
GRIN2A Q12879 2/20 0.51
GRIN2B Q13224 2/20 0.51
GRIN2C Q14957 1/20 0.51
MAPT P10636 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 2/20 0.48
BCHE P06276 1/20 0.48
LMNA P02545 6/20 0.47
ALOX15 P16050 1/20 0.45
EPHX2 P34913 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
MAPK1 P28482 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5503332 0.81 AR (0.63) ARALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL5114895 0.73 PTGDR2 (0.61)
SCHEMBL5503450 0.73 AR (0.63) ARALDH1A1GRIN2AGRIN2BGRIN2C
SCHEMBL14304932 0.71 BCHE (0.86) ARALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL9514166 0.71 ALDH1A1 (1.00) ARALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL14303261 0.70 BCHE (0.83) ARALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL14304381 0.70 BCHE (0.83) ARALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL6141660 0.70 BCHE (0.83) ARALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL14303260 0.70 BCHE (0.83) ARALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL14304387 0.70 BCHE (0.83) ARALDH1A1MAPTSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784182-A1 2-SULFANYL-BENZIMIDAZOL-1-YL-ACETIC ACID DERIVATIVES AS CRTH2 ANTAGONISTS Actelion Pharmaceuticals Ltd. (CH) 2007-05-16 EP claimed
WO-2006021418-A1 2-SULFANYL-BENZOIMIDAZOL-1-YL-ACETIC ACID DERIVATIVES AS CRTH2 ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-02 WO claimed