SCHEMBL5500282

SCHEMBL5500282

CCCn1c(=O)c2[nH]c(C3CC4CC(=CC(=O)O)C3C4)nc2n(CCC)c1=O

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 10/20 0.62
ADORA2A P29274 6/20 0.54
ADORA2B P29275 5/20 0.54
MEN1 O00255 1/20 0.54
GMNN O75496 1/20 0.54
LMNA P02545 1/20 0.54
CYP1A2 P05177 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
TSHR P16473 1/20 0.54
PMP22 Q01453 1/20 0.54
KMT2A Q03164 1/20 0.54
HIF1A Q16665 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7644015 0.82 ADORA1 (0.71) ADORA1ADORA2AADORA2BMEN1GMNN
SCHEMBL4990267 0.82 ADORA1 (0.60) ADORA1ADORA2AADORA2BMEN1GMNN
SCHEMBL5201345 0.82 ADORA1 (0.60) ADORA1ADORA2AADORA2BMEN1GMNN
SCHEMBL5004424 0.77 ADORA1 (0.59) ADORA1ADORA2AADORA2BMEN1GMNN
SCHEMBL5004423 0.77 ADORA1 (0.59) ADORA1ADORA2AADORA2BMEN1GMNN
SCHEMBL4985610 0.77 ADORA1 (0.65) ADORA1ADORA2AADORA2BMEN1GMNN
SCHEMBL3686177 0.76 ADORA1 (0.68) ADORA1ADORA2AADORA2BMEN1GMNN
SCHEMBL7431499 0.75 ADORA1 (0.70) ADORA1ADORA2AADORA2BMEN1GMNN
SCHEMBL7439146 0.75 ADORA1 (0.70) ADORA1ADORA2AADORA2BMEN1GMNN
SCHEMBL5498012 0.75 ADORA1 (0.61) ADORA1ADORA2AADORA2BMEN1GMNN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230241-B1 ADENOSINE RECEPTOR ANTAGONISTS AND METHODS OF MAKING AND USING THE SAME BIOGEN IDEC INC (US) 2007-02-07 EP disclosed