SCHEMBL5501024

SCHEMBL5501024

Cc1ccc(S(=O)(=O)OCC2CCN(C(=O)O)C[C@@H]2O)cc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.44
CYP1A2 P05177 1/20 0.44
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
STAT3 P40763 1/20 0.39
KMT2A Q03164 2/20 0.39
CYP46A1 Q9Y6A2 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3021790 1.00 CYP2D6 (0.44) CYP2D6CYP1A2ALDH1A1KDM4ELMNA
SCHEMBL3021792 1.00 CYP2D6 (0.44) CYP2D6CYP1A2ALDH1A1KDM4ELMNA
SCHEMBL3021789 1.00 CYP2D6 (0.44) CYP2D6CYP1A2ALDH1A1KDM4ELMNA
SCHEMBL26906971 0.89 STAT3 (0.41) CYP2D6CYP1A2ALDH1A1KDM4ELMNA
SCHEMBL505550 0.85 GPR119 (0.48) KMT2A
SCHEMBL856350 0.85 GPR119 (0.48) KMT2A
SCHEMBL857313 0.85 GPR119 (0.48) KMT2A
SCHEMBL856351 0.85 GPR119 (0.48) KMT2A
SCHEMBL29895401 0.85 GPR119 (0.48) KMT2A
SCHEMBL856352 0.85 GPR119 (0.48) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641784-B1 4-(AMINOMETHYL)-PIPERIDINE BENZAMIDES AS 5HT4 -ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2007-06-13 EP disclosed
EP-1641784-A1 4-(AMINOMETHYL)-PIPERIDINE BENZAMIDES AS 5HT4 -ANTAGONISTS JANSSEN PHARMACEUTICA N.V. (BE) 2006-04-05 EP disclosed
WO-2005000838-A1 4-(AMINOMETHYL)-PIPERIDINE BENZAMIDES AS 5HT4-ANTAGONISTS JANSSEN PHARMACEUTICA N.V. (BE) 2005-01-06 WO disclosed