Ethalfluralin

Ethalfluralin

SCHEMBL55014

C=C(C)CN(CC)c1c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.64
MAPK1 P28482 3/20 0.64
MAPT P10636 3/20 0.64
TDP1 Q9NUW8 3/20 0.63
TSHR P16473 2/20 0.63
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
HIF1A Q16665 1/20 0.44
TXNRD1 Q16881 1/20 0.44
TXNRD3 Q86VQ6 1/20 0.44
TXNRD2 Q9NNW7 1/20 0.44
GAA P10253 2/20 0.42
LMNA P02545 1/20 0.42
HPD P32754 1/20 0.40
HCAR3 P49019 1/20 0.39
PTPN5 P54829 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethalfluralin SCHEMBL4899703 1.00 CYP3A4 (0.64) CYP3A4MAPK1MAPTTDP1TSHR
SCHEMBL9451050 0.90 TDP1 (0.76) CYP3A4MAPK1MAPTTDP1TSHR
SCHEMBL135804 0.90 TDP1 (0.76) CYP3A4MAPK1MAPTTDP1TSHR
SCHEMBL8857960 0.88 CYP3A4 (0.63) CYP3A4MAPK1MAPTTDP1TSHR
SCHEMBL11203878 0.86 CYP3A4 (0.78) CYP3A4MAPK1MAPTTDP1TSHR
SCHEMBL10867828 0.85 MAPK1 (0.46) CYP3A4MAPK1MAPTTDP1TSHR
Isopropalin SCHEMBL17555757 0.82 TDP1 (0.67) CYP3A4MAPK1MAPTTDP1TSHR
SCHEMBL11204357 0.81 TDP1 (0.89) CYP3A4MAPK1MAPTTDP1TSHR
SCHEMBL11513263 0.81 TDP1 (0.51) CYP3A4MAPK1MAPTTDP1TSHR
SCHEMBL11205360 0.80 CYP3A4 (0.66) CYP3A4MAPK1MAPTTDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 15732 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144260-A1 COMPOSITION AND METHOD FOR IMPROVING AGRONOMIC TRAITS OF A PLANT THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2026-05-28 US claimed
US-20260096553-A1 MICROENCAPSULATED HERBICIDES MONSANTO TECHNOLOGY LLC (US) 2026-04-09 US claimed
US-20260060254-A1 HERBICIDAL COMPOSITIONS BAYER AG (DE) 2026-03-05 US claimed
US-20260020563-A1 METHOD FOR CONTROLLING PESTS OF FARM CROPS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2026-01-22 US claimed
US-20260007133-A1 HERBICIDAL COMPOSITION COMPRISING AZINE COMPOUNDS BASF SE (DE) 2026-01-08 US claimed
US-20250374926-A1 NOVEL DERIVATIVES OF NON-CODED AMINO ACIDS AND THEIR USE IN CROP PROTECTION FORTEPHEST LTD. (IL) 2025-12-11 US claimed
US-20250366479-A1 Non-Aqueous Organo Liquid Delivery Systems containing dispersed Organo Polycarboxylate Functionalities that improves efficiencies and properties of nitrogen sources SOILGENIC TECH LLC (US) 2025-12-04 US claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-4646109-A2 NATURAL LIPID PARTICLE FORMULATIONS FOR AGRICULTURAL APPLICATIONS Invaio Sciences, Inc. (US) 2025-11-12 EP claimed
EP-0126591-B1 DINITROANILINE COMPOSITIONS STABILIZED BY INCORPORATION OF ADDITION COMPOUND OF BISULFITE AND ALDEHYDE OR KETONE ELI LILLY AND COMPANY (US) 1987-04-08 EP claimed
EP-0200935-A2 Synergistic herbicidal compositions STAUFFER CHEMICAL COMPANY (US) 1986-11-12 EP claimed
US-4501608-A STABILIZING DINITROANILINE HERBICIDES BY ADDING A BISULFITE COMPOUND AND AN ALDEHYDE OR KETONE ELI LILLY AND COMPANY (US) 1985-02-26 US claimed
EP-0126591-A1 Dinitroaniline compositions stabilized by incorporation of addition compound of bisulfite and aldehyde or ketone ELI LILLY AND COMPANY (US) 1984-11-28 EP claimed
EP-0124993-A1 Granular herbicidal formulations ELI LILLY AND COMPANY (US) 1984-11-14 EP claimed
EP-0070219-B1 HERBICIDAL COMPOSITIONS BASED ON 4-AMINO-6-CHLORO-5-ALKYLTHIOPYRIMIDINE DERIVATIVES AND 2,6-DINITROANILINE DERIVATIVES, AND METHOD OF TREATING CROPS WITH SAID COMPOSITIONS P C U K PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1984-10-24 EP claimed
EP-0070130-A1 Improvement in or relating to benzoylphenyl urea derivatives ELI LILLY AND COMPANY (US) 1983-01-19 EP claimed
US-4226789-A Removal of nitrosamines from denitroanilines by treatment with HCl ELI LILLY AND COMPANY (US) 1980-10-07 US claimed
US-4185035-A REMOVAL OF NITROSAMINES WITH PHOSPHORUS HALIDES ELI LILLY AND COMPANY (US) 1980-01-22 US claimed
EP-0005917-A1 Herbicidal method and mixtures of herbicidal heterocyclic compounds FISONS plc (GB) 1979-12-12 EP claimed