SCHEMBL5501933

SCHEMBL5501933

COc1cccc(-c2n[nH]c(N)c2C#N)c1

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.64
ADORA2A P29274 5/20 0.64
HPGD P15428 2/20 0.64
HTT P42858 2/20 0.64
ADORA2B P29275 2/20 0.64
TP53 P04637 1/20 0.64
RXFP1 Q9HBX9 2/20 0.58
MAPT P10636 1/20 0.58
NPSR1 Q6W5P4 2/20 0.54
KMT2A Q03164 2/20 0.54
MEN1 O00255 1/20 0.54
GAA P10253 1/20 0.52
PLA2G2A P14555 1/20 0.50
KDM4E B2RXH2 3/20 0.49
GLA P06280 1/20 0.49
MKNK1 Q9BUB5 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
DCUN1D1 Q96GG9 1/20 0.48
SQOR Q9Y6N5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18866750 0.84 ADORA2A (0.52) ADORA1ADORA2AHPGDHTTADORA2B
SCHEMBL15214874 0.82 ADORA1 (0.50) ADORA1ADORA2AHPGDHTTADORA2B
SCHEMBL8124145 0.82 ADORA1 (0.65) ADORA1ADORA2AHPGDADORA2BMAPT
SCHEMBL23998166 0.81 ADORA2A (0.58) ADORA1ADORA2AHPGDHTTADORA2B
SCHEMBL30250859 0.81 ADORA2A (0.58) ADORA1ADORA2AHPGDHTTADORA2B
SCHEMBL10360609 0.79 ATM (0.44) ADORA1ADORA2AHPGDHTTADORA2B
SCHEMBL3614512 0.79 ADORA1 (0.47) ADORA1ADORA2AHPGDHTTADORA2B
SCHEMBL2645516 0.78 ADORA1 (0.58) ADORA1ADORA2AHPGDADORA2BKMT2A
SCHEMBL15286427 0.77 ADORA1 (0.67) ADORA1ADORA2AHPGDHTTADORA2B
SCHEMBL15286448 0.77 ADORA1 (0.67) ADORA1ADORA2AHPGDHTTADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778718-A1 INHIBITORS OF IAP Genentech, Inc. (US) 2007-05-02 EP disclosed
WO-2006014361-A1 INHIBITORS OF IAP GENENTECH, INC. (US) 2006-02-09 WO disclosed