SCHEMBL15214874

SCHEMBL15214874

Cc1cccc(-c2n[nH]c(N)c2C#N)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.50
ADORA2A P29274 5/20 0.50
ATM Q13315 1/20 0.47
HTR7 P34969 1/20 0.45
HPGD P15428 3/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ADORA2B P29275 3/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
POLB P06746 1/20 0.43
TP53 P04637 1/20 0.43
HTT P42858 1/20 0.43
LRRK2 Q5S007 1/20 0.42
RAB9A P51151 1/20 0.41
GAA P10253 1/20 0.41
GFER P55789 1/20 0.41
PIK3CD O00329 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30250859 0.83 ADORA2A (0.58) ADORA1ADORA2AATMHPGDADORA2B
SCHEMBL23998166 0.83 ADORA2A (0.58) ADORA1ADORA2AATMHPGDADORA2B
SCHEMBL5501933 0.82 ADORA1 (0.64) ADORA1ADORA2AHPGDKDM4EADORA2B
SCHEMBL10360609 0.81 ATM (0.44) ADORA1ADORA2AATMHPGDADORA2B
SCHEMBL8914694 0.81 ADORA1 (0.54) ADORA1ADORA2AHPGDALDH1A1KDM4E
SCHEMBL2645516 0.80 ADORA1 (0.58) ADORA1ADORA2AHPGDALDH1A1KDM4E
SCHEMBL18866750 0.78 ADORA2A (0.52) ADORA1ADORA2AHPGDALDH1A1ADORA2B
SCHEMBL5501424 0.76 LMNA (0.54) ATMHPGDALDH1A1MEN1KMT2A
SCHEMBL8130126 0.74 GAA (0.65) HPGDKDM4EKMT2ARAB9AGAA
SCHEMBL14809869 0.74 ADORA2A (0.58) ADORA1ADORA2AKDM4EADORA2BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9067928-B2 Compounds and methods of use ABBVIE INC. (US) 2015-06-30 US disclosed
US-8518970-B2 Compounds and methods of use ABBVIE INC. (US) 2013-08-27 US disclosed