SCHEMBL5503067

SCHEMBL5503067

CC1(C)O[C@@H]2[C@H](O1)[C@@H](CO)O[C@H]2n1cnc2c(NC3CCCCC3)nc(F)nc21

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.57
ADORA2A P29274 3/20 0.57
ADORA2B P29275 2/20 0.57
ADORA1 P30542 2/20 0.57
MEN1 O00255 1/20 0.57
CYP1A2 P05177 1/20 0.57
MAPK1 P28482 1/20 0.57
KMT2A Q03164 1/20 0.57
RXFP1 Q9HBX9 1/20 0.56
ALOX15 P16050 1/20 0.54
PI4KA P42356 1/20 0.52
PI4K2B Q8TCG2 1/20 0.52
PI4K2A Q9BTU6 1/20 0.52
PI4KB Q9UBF8 1/20 0.52
PMP22 Q01453 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
TDP1 Q9NUW8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20180024 0.89 ADORA3 (0.72) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL5511103 0.88 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL5508361 0.86 TSHR (0.70) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL5507191 0.85 ADORA3 (0.69) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL12200089 0.85 ADORA3 (0.69) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL15144301 0.85 ADORA3 (0.69) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL7735031 0.85 ADORA3 (0.69) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL5509724 0.85 ADORA3 (0.46) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL6574020 0.82 ADORA3 (0.66) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL4649323 0.82 PI4KA (0.68) ADORA3ADORA2AADORA2BADORA1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537133-B1 PARTIAL AND FULL AGONISTS OF A1 ADENOSINE RECEPTORS CV THERAPEUTICS INC (US) 2007-07-25 EP disclosed